The Chalcogen Or The Acyclic Nitrogen Is Bonded Directly To The Six Membered Hetero Ring Patents (Class 546/292)
  • Patent number: 4375546
    Abstract: Substituted pyridinols are reacted with an isocyanatoethyl alkanoate in an inert solvent in the presence of an activating agent to form a group of biologically active organic compounds. These compounds are useful as broad spectrum herbicides effective against a variety of grassy weeds, broadleaf weeds and grassy crops. Compounds of this invention may also be utilized as fungicides.
    Type: Grant
    Filed: November 16, 1981
    Date of Patent: March 1, 1983
    Assignee: The Dow Chemical Company
    Inventor: Chester E. Pawloski
  • Patent number: 4372778
    Abstract: N-(Pyridinylaminocarbonyl)benzenesulfonamides are useful for the regulation of plant growth and as pre-emergence and post-emergence herbicides.
    Type: Grant
    Filed: May 29, 1981
    Date of Patent: February 8, 1983
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: George Levitt
  • Patent number: 4358606
    Abstract: Novel esters of phenylalkyloxy- or phenylalkylthioacylamino acids and pyridylalkyloxy- or pyridylalkylthioacylamino acids, synthesis thereof, intermediates therefor, and the use of said esters for the control of weeds.
    Type: Grant
    Filed: June 19, 1981
    Date of Patent: November 9, 1982
    Assignee: Zoecon Corporation
    Inventors: Shy-Fuh Lee, Clive A. Henrick
  • Patent number: 4344893
    Abstract: Novel compounds are described which are substituted benzophenone hydrazones. They have pesticidal activity, especially against insects and acarids, and pesticidal compositions and methods are described. Methods of making the compounds, and novel intermediates, are also described.
    Type: Grant
    Filed: February 25, 1980
    Date of Patent: August 17, 1982
    Assignee: The Boots Company Limited
    Inventors: Leonard G. Copping, John C. Kerry, Thomas I. Watkins, Robert J. Willis, Bryan H. Palmer
  • Patent number: 4308054
    Abstract: N-(2,6-disubstituted 4-pyridyl)-N'-phenylurea compounds are plant growth regulators having potent cytokinin activity. N-(2,6-dichloro-4-pyridyl)-N'-phenylurea is useful for regulating plant growth.
    Type: Grant
    Filed: October 24, 1980
    Date of Patent: December 29, 1981
    Inventors: Yo Isogai, Soshiro Takahashi, Koichi Shudo, Toshihiko Okamoto
  • Patent number: 4293330
    Abstract: N-(Pyridinylaminocarbonyl)benzenesulfonamides are useful for the regulation of plant growth and as pre-emergence and post-emergence herbicides.
    Type: Grant
    Filed: September 29, 1980
    Date of Patent: October 6, 1981
    Assignee: E. I. Du Pont de Nemours and Company
    Inventor: George Levitt
  • Patent number: 4279639
    Abstract: Plant growth and suppression regulators of the N-(2-substituted-4-pyridyl)urea and thiourea type are provided, which exhibit excellent cytokinin-like activities and are thus useful for regulating plant growth in various fashions, such as acceleration of growth when used in flowering or fruiting at a controlled time when used in small amounts, and controlling compositions such as sugar, alkaloids, etc. of plants, or suppression of plant growth when used in an amount higher than optimal for growth acceleration, etc.
    Type: Grant
    Filed: August 1, 1979
    Date of Patent: July 21, 1981
    Assignees: Toshihiko Okamoto, Yo Isogai, Koichi Shudo, Susumu Sato
    Inventors: Toshihiko Okamoto, Yo Isogai, Koichi Shudo, Soshiro Takahashi
  • Patent number: 4264605
    Abstract: The present invention is directed to 1-benzoyl-3-(aryloxy- or arylthio-pyridinyl)urea compounds useful as insecticides.
    Type: Grant
    Filed: June 13, 1979
    Date of Patent: April 28, 1981
    Assignee: Eli Lilly and Company
    Inventors: Robert G. Suhr, John L. Miesel
  • Patent number: 4261730
    Abstract: Aromatic acids having the following formula ##STR1## have been found to be effective plant growth regulants especially for the treatment of corn plants.
    Type: Grant
    Filed: August 9, 1978
    Date of Patent: April 14, 1981
    Assignee: Monsanto Company
    Inventors: Frederic G. Bollinger, John J. D'Amico, Dale J. Hansen
  • Patent number: 4260410
    Abstract: Novel N-haloacetylphenylamino carbonyl oximes represented by the formula ##STR1## wherein Ar is phenyl or substituted phenyl; R.sup.1 is halomethyl; R.sup.2 and R.sup.3 are each independently hydrogen, alkyl, phenyl, benzyl, substituted phenyl or benzyl, haloalkyl, cyanoalkyl, alkoxyalkyl, alkylthioalkyl or thiocyanoalkyl; R.sup.4 is hydrogen or alkyl; n is 0 or 1; m is 0 or 1; R is hydrogen, alkyl, alkenyl, alkynyl, alkylthioalkyl, haloalkyl, alkoxyalkyl, cyanoalkyl, phenyl, benzyl, substituted phenyl or benzyl, or R is acyl of the formula ##STR2## wherein R.sup.5 is hydrogen, alkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl, alkoxy, alkylthio, acetonyl, or the group -NR'R" wherein R' and R" are independently hydrogen, alkyl or phenyl; with the proviso that R.sup.2 and R.sup.3 may be joined together to form a carbocyclic ring or a heterocyclic ring; or R and R.sup.2 may be joined together to form a heterocyclic ring; or R and R.sup.3 may be joined together to form a heterocyclic ring.
    Type: Grant
    Filed: February 23, 1979
    Date of Patent: April 7, 1981
    Assignee: Chevron Research Company
    Inventors: William L. Schinski, David C. K. Chan, Irene C. Huang
  • Patent number: 4252813
    Abstract: Compounds of the formula ##STR1## are useful as anti-allergy agents.
    Type: Grant
    Filed: November 19, 1979
    Date of Patent: February 24, 1981
    Assignee: The Upjohn Company
    Inventor: John B. Wright
  • Patent number: 4241068
    Abstract: Compounds of the formula ##STR1## wherein A is .dbd.CH-- or .dbd.N--;R.sub.1 is (a) hydrogen, lower alkyl, lower alkoxy or a fused benzene ring, or (b) --CO--R.sub.4, tetrazol-5-yl or cyano in the 4- or 5-position;R.sub.2 is --CO--R.sub.4, tetrazol-5-yl, cyano or, when R.sub.1 has one of the meanings included in (b), also hydrogen, lower alkyl, lower alkoxy or a fused benzene ring;R.sub.3 is hydrogen or lower alkanoyl; andR.sub.4 is hydroxyl, amino, hydroxy-amino, tetrazol-5-yl-amino or lower alkoxy;internal salts thereof, and non-toxic salts thereof formed with a basic substance. The compounds as well as their salts are useful as antiallergics.
    Type: Grant
    Filed: August 7, 1979
    Date of Patent: December 23, 1980
    Assignee: Boehringer Ingelheim GmbH
    Inventors: Kurt Schromm, Anton Mentrup, Ernst-Otto Renth, Armin Fugner, Volker Jacobi
  • Patent number: 4203988
    Abstract: Compounds of the formula ##STR1## have been found to inhibit gastric secretion in mammalian species.
    Type: Grant
    Filed: September 18, 1978
    Date of Patent: May 20, 1980
    Assignee: Merck & Co., Inc.
    Inventors: William A. Bolhofer, Edward J. Cragoe, Jr., Jacob M. Hoffman, Jr.
  • Patent number: 4181658
    Abstract: Benzoic acid derivatives of the formula ##STR1## wherein T is hydrogen or halogen, W is a carboxyl group, an ester or salt thereof; X is ##STR2## wherein R.sub.1 is alkyl having from 2 to 8 carbon atoms, aralkyl or phenyl, cycloalkyl, cycloalkylalkyl or alkylcycloalkyl; R.sub.2 is hydrogen or halogen, R.sub.3 is alkyl having from 5 to 8 carbon atoms, aralkyl or phenyl, or cycloalkyl having from 5 to 8 carbon atoms; R.sub.4 is hydrogen or alkyl; Y is a single chemical bond or a hydrocarbon chain having from 1 to 3 carbon atoms; and Z is hydrogen, halogen, alkyl, alkoxy, alkoxyalkoxy or alkenyloxy, have a blood sugar lowering effect and can be used for the treatment of Diabetes mellitus.
    Type: Grant
    Filed: February 16, 1978
    Date of Patent: January 1, 1980
    Assignee: Hoechst Aktiengesellschaft
    Inventors: Volker Hitzel, Rudi Weyer, Karl Geisen, Werner Pfaff
  • Patent number: 4174210
    Abstract: Novel N-haloacetylphenylamino carbonyl oximes represented by the formula ##STR1## wherein Ar is aryl, R.sup.1 is halomethyl, R.sup.2 is hydrogen, alkyl or aryl, R.sup.3 is hydrogen, alkyl or aryl, n is 0 or 1 and R is hydrogen, aryl, alkyl, alkenyl or alkynyl, with the proviso that R.sup.2 and R.sup.3 may be joined together to form a carbocyclic ring of 5 to 6 carbon atoms or a heterocyclic ring of one N, O or S hetero atom and 4 to 5 carbon atoms. The oxime compounds are useful as herbicides and plant growth regulators.
    Type: Grant
    Filed: March 31, 1978
    Date of Patent: November 13, 1979
    Assignee: Chevron Research Company
    Inventors: William L. Schinski, Irene C. Huang, David C. K. Chan
  • Patent number: 4173639
    Abstract: The present invention is directed to 1-benzoyl-3-(alkoxy- or alkylthiopyridinyl)urea compounds useful as insecticides.
    Type: Grant
    Filed: August 31, 1978
    Date of Patent: November 6, 1979
    Assignee: Eli Lilly and Company
    Inventor: Robert G. Suhr
  • Patent number: 4149872
    Abstract: Compounds of the formula ##STR1## wherein A is ##STR2## in which R.sup.1 is alkyl and n is 0-1, or ##STR3## in which R.sup.2 is hydrogen, alkyl or halogen; Y is halogen or alkyl; and X is halogen, --NR.sup.3 R.sup.4 in which R.sup.3 and R.sup.4 each independently is hydrogen or alkyl; OR.sup.5 ; SR.sup.5 ; S(O)R.sup.5 or S(O).sub.2 R.sup.5, in which R.sup.5 is alkyl, are useful as herbicides.
    Type: Grant
    Filed: July 21, 1977
    Date of Patent: April 17, 1979
    Assignee: Shell Oil Company
    Inventor: Kurt H. G. Pilgram
  • Patent number: 4139537
    Abstract: Cardiac arrhythmias can be treated by administering an effective amount of 3-aryloxy-1-(2-or 4-iminodihydro-1-pyridyl)-2-propanol or phamaceutically acceptable acid addition compound. Many new effective compounds of this type are disclosed.
    Type: Grant
    Filed: June 29, 1976
    Date of Patent: February 13, 1979
    Assignee: Cooper Laboratories, Inc.
    Inventors: Julius Diamond, Ronald A. Wohl