Publication number: 20110009428
Abstract: The compounds of the subject invention have a structure according to formula I: wherein X is S or SO2; R1 is (1C-6C)alkyl, (3C-6C)alkenyl, or (3C-6C)alkynyl, each optionally substituted with (3C-6C)cycloalkyl, OH, OC(O)(1C-4C)alkyl, (1C-4C)alkoxy, halogen, cyano, formyl, C(O)(1C-4C)alkyl, CO2H, CO2(1C-4C)alkyl, C(O)NR5R6, S(O)(1C-4C)alkyl or S(O)2(1C-4C)alkyl; R2 is hydrogen, (1C-4C)alkyl or C(O)(1C-4C)alkyl; R3 is a phenyl group optionally substituted with (1C-4C)alkyl, (1C-4C)fluoroalkyl, (1C-4C)alkoxy, (1C-4C)fluoroalkoxy, halogen, cyano or nitro; or R3 is a 5- or 6-membered aromatic heterocyclic ring structure optionally substituted with (1C-4C)alkyl, (1C-4C)fluoroalkyl, (1C-4C)alkoxy, halogen or cyano; R4 is a phenyl group or an aromatic 6-membered heterocycle, substituted at the ortho position with 1-hydroxy(1C-4C)alkyl, (1C-4C)alkoxy, C(O)(1C-4C)alkyl, CO2(1C-4C)alkyl, C(O)NH2, cyano, nitro, or CH?NOR7, and optionally further substituted with (1C-2C)alkyl, (1C-2C)fluoroalkyl or halogen; or R4
Type:
Application
Filed:
September 22, 2010
Publication date:
January 13, 2011
Applicant:
N.V. Organon
Inventors:
Jaap Van Der Louw, Neeltje Miranda Teerhuis, Johannes Petrus Maria Lommerse, Herman Thijs Stock, Pedro Harold Han Hermkens
Patent number: 7812041
Abstract: The present invention relates to compounds of the general formula (I) and salts and physiologically functional derivatives thereof, wherein R1 is independently hydrogen; alkyl, cycloalkyl, hydroxyalkyl, haloalkyl, haloalkyloxy, aryl, substituted aryl, heteroaryl, substituted heteroaryl, arylalkyl or substituted arylalkyl; R2 is independently —NR3R4, R3 is independently alkyl, cycloalkyl, alkoxy, alkylamine, —OH, —SH, alkylthio, hydroxyalkyl, haloalkyl, haloalkyloxy, aryl or heteroaryl, R4 is independently alkyl, cycloalkyl, alkoxy, alkylamine, alkylthio, hydroxyalkyl, haloalkyl, haloalkyloxy, aryl or heteroaryl; R5 is independently H, COR6, CO2R6, SOR6, SO3R6, alkyl, cycloalkyl, alkoxy, —NH2, alkylamine, —NR7COR6, halogen, —OH, —SH, alkylthio, hydroxyalkyl, haloalkyl, haloalkyloxy, aryl or heteroaryl; R6 is independently H, alkyl, cycloalkyl, —NH2, alkylamine, aryl or heteroaryl; R7 is independently H, alkyl, cycloalkyl, alkoxy, —OH, —SH, alkylthio, hydroxyalkyl, aryl, or heteroaryl; p is 0, or 1;
Type:
Grant
Filed:
July 29, 2005
Date of Patent:
October 12, 2010
Assignee:
4SC AG
Inventors:
Johann Leban, Harald Schmitt, Kristina Wolf, Stefano Pegoraro, Andreas Wuzik
Patent number: 7696129
Abstract: The present invention provides a substituted anilide derivative of formula (I): {wherein Z is a group of formula (II) or (III) (in these formulas, A is C1-C6 alkylene, C2-C6 alkenylene, etc., R1 is H, halogen, —C(R5)?NOR6, (substituted) phenyl, (substituted) heterocyclic ring, -A1-R7, etc.; R2 is H, C1-C4 alkyl, etc.), R3 is H, C1-C4 alkyl, etc.; R4 is H, F, fluoro C1-C6 alkyl; Rf is F, fluoro C1-C6 alkyl; 1 is 0 to 2; Y is halogen, (substituted) phenyl, (substituted) phenoxy, etc.; and m is 0 to 3}, an intermediate thereof, an agrohorticultural agent, and a method for the use thereof. The compound of the present invention exhibits, at a low dosage, high uptake and translocation from the root and an excellent insecticidal effect especially when applied to soil.
Type:
Grant
Filed:
May 16, 2002
Date of Patent:
April 13, 2010
Assignee:
Nihon Nohyaku Co., Ltd.
Inventors:
Makoto Goto, Minoru Yamaguchi, Hiroto Harayama, Hayami Nakao, Takashi Furuya, Masanori Tohnishi, Masayuki Morimoto, Shinsuke Fujioka