1,3,5-triazine Ring Patents (Class 544/113)
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Patent number: 4565815Abstract: A compound having anti-ulcer activity and having the formula ##STR1## wherein D is H, SH, NH.sub.2, OH, R.sup.4 S where R.sup.4 is a lower alkyl group; E is OH or NH.sub.2 ; J is H or aryl; X is CH or N; Y is CH, N, or CT, wherein T is a halogen; Z is CH or N; A is ##STR2## and replaces a hydrogen of D, X, or E; R.sup.1 is H or CH.sub.3 ; L is CH.sub.2 S; Q is O or CH.sub.2 S; n is 0 or 1; 2 m 4; each R.sup.2 and R.sup.3, independently, is H, lower alkyl, cycloalkyl, or arylalkyl; or R.sup.2 and R.sup.3, together with the nitrogen atom to which they are attached, form a 4, 5, or 6 membered heterocyclic ring containing 0, 1, or 2 oxygen atoms and 1, 2, or 3 nitrogen atoms and being unsubstituted or lower alkyl substituted; or a pharmaceutically acceptable salt thereof.Type: GrantFiled: May 25, 1984Date of Patent: January 21, 1986Assignee: Biomeasure, Inc.Inventors: Sun H. Kim, Jacques-Pierre Moreau
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Patent number: 4562188Abstract: A method for the treatment of irritable bowel syndrome using a 1,3,5-triazin-2-one and a class of 6-amino and 6-mercaptyl-1,3,5-triazin-2-one compounds.Type: GrantFiled: January 13, 1984Date of Patent: December 31, 1985Assignee: William H. Rorer, Inc.Inventors: Donald E. Kuhla, William L. Studt, Henry F. Campbell, John Yelnosky
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Patent number: 4547548Abstract: Polycondensation compounds containing piperidine and triazine groups, having a mean molecular weight from 1000 to 20,000 and constituted by structural units a and b of the formula ##STR1## are suitable as anti-actinic stabilizers for incorporation in polymeric materials.Type: GrantFiled: July 19, 1984Date of Patent: October 15, 1985Assignee: Ciba-Geigy S.p.A.Inventor: Giuseppe Cantatore
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Patent number: 4521597Abstract: A novel process for producing sulfonylureas of the formula I having a herbicidal action and an action regulating plant growth ##STR1## wherein A is an unsubstituted or substituted phenyl, naphthyl, furan, thiophene or pyridine group, E is a nitrogen atom or the methine group, R.sub.a is hydrogen, halogen, C.sub.1 -C.sub.5 -alkyl, C.sub.1 -C.sub.5 -haloalkyl, C.sub.1 -C.sub.5 -alkoxy, C.sub.1 -C.sub.5 -haloalkoxy, C.sub.1 -C.sub.5 -alkylthio or C.sub.2 -C.sub.10 -alkoxyalkoxy, and R.sub.b is the same as R.sub.Type: GrantFiled: October 14, 1983Date of Patent: June 4, 1985Assignee: Ciba Geigy CorporationInventors: Haukur Kristinsson, Werner Topfl
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Patent number: 4500710Abstract: Quinophthalone dyes for cellulose-containing fibers represented by the following general formula: ##STR1## wherein X represents a hydrogen atom, a chlorine atom or a bromine atom, --A-- represents a methylene group, an ethylene group, a propylene group or a 1,3-butylene group, n represents 0 or 1, --Y-- represents a linkage group of --O-- or --S--, R.sup.1 and R.sup.2 each represents a hydrogen atom, an alkyl or alkenyl group which may optionally be substituted with a cyano group, a hydroxy group, a lower alkoxy group or by a dialkylamino group, or R.sup.1 and R.sup.2 may be combined together with the adjacent nitrogen atom to form a 5- or 6-membered, nitrogen-containing heterocyclic ring having the total carbon atom number in R.sup.1 and R.sup.2 of up to 18.Type: GrantFiled: June 16, 1983Date of Patent: February 19, 1985Assignee: Mitsubishi Chemical Industries, LimitedInventors: Toshio Niwa, Toshio Hihara
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Patent number: 4496564Abstract: The invention relates to amide derivatives which are histamine H-2 antagonists and which inhibit gastric acid secretion. According to the invention there is provided a guanidine derivative of the formula I: ##STR1## in which R.sup.1 is a hydrogen or 1-10C alkyl, 3-8C cycloalkyl, 4-14C cycloalkylalkyl, 3-6C alkenyl, 3-6C alkynyl, 1-6C alkanoyl, 6-10C aryl, 7-11C aralkyl or 7-11C aroyl, the aryl, aralkyl and aroyl radical being optionally substituted; ring X is a heterocyclic ring as defined in the specification; A is phenylene or 5-7C cycloalkylene, or a 1-8C alkylene into which is optionally inserted one or two groups; D is O or S; and R.sup.2 and R.sup.3 are hydrogen or a variety of radicals described in the specification: and the pharmaceutically-acceptable acid-addition salts thereof. Manufacturing processes and pharmaceutical compositions are also described.Type: GrantFiled: March 1, 1982Date of Patent: January 29, 1985Assignees: ICI Americas Inc., Imperial Chemical Industries PLCInventors: Tobias O. Yellin, David J. Gilman
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Patent number: 4496726Abstract: Hitherto unknown polyalkylpiperidinylaminotriazines having a structure of the type ##STR1## are obtained from halogenotriazinyl compounds and aminoethylaminoethanols and can be converted into further derivatives with isocyanates, esters and acid chlorides to give new stabilizers for polymers, which stabilizers are distinguished by very good migration resistance.Type: GrantFiled: August 2, 1982Date of Patent: January 29, 1985Inventors: Hartmut Wiezer, Gerhard Pfahler
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Patent number: 4492599Abstract: This invention relates to novel urea and isourea compounds, agricultural compositions containing them and to their method of use as pre- and post- emergence herbicides and to plant growth regulants.Type: GrantFiled: September 27, 1982Date of Patent: January 8, 1985Assignee: E. I. Du Pont de Nemours and CompanyInventors: George Levitt, Wallace C. Petersen
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Patent number: 4486589Abstract: N-(heterocyclicaminocarbonyl)-ortho-haloalkylbenzenesulfonamides, such as 2-(dichloromethyl)-N-[(4-methoxy-6-methylprimidin-2-yl) aminocarbonyl]-benzenesulfonamide, are useful as preemergent or postemergent herbicides or as plant growth regulants.Type: GrantFiled: October 21, 1982Date of Patent: December 4, 1984Assignee: E. I. Du Pont de Nemours and CompanyInventor: William B. Farnham
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Patent number: 4483857Abstract: 2,4-Diaminoquinazoline compounds of the formula ##STR1## or a pharmaceutically acceptable salt thereof wherein R is a pyrimidinyl, pyrazinyl, pyridazinyl or triazinyl group linked to the piperazine ring by one of its carbon atoms, and optionally substituted by hydroxy, halogen, alkyl, aralkyl, alkoxy, aralkoxy, alkylthio, aryl, aryloxy and certain amino groups; their use as an antihypertensive agent and pharmaceutical compositions containing them.Type: GrantFiled: August 24, 1983Date of Patent: November 20, 1984Assignee: Pfizer Inc.Inventors: Simon F. Campbell, Rhona M. Plews
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Patent number: 4481029Abstract: This invention relates to ureas and isoureas which are useful as herbicides and plant growth regulants. In particular, compounds of the instant invention have demonstrated great selectivity.Type: GrantFiled: December 16, 1982Date of Patent: November 6, 1984Assignee: E. I. Du Pont de Nemours and CompanyInventor: George Levitt
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Patent number: 4480092Abstract: A branched chain polyalkylenepolyamine ("PAPA") amine having plural amine groups including a secondary amine group intermediate terminal primary amine groups and having at least two carbon atoms between each amine group, is reductively alkylated with a ketone to provide a PAPA alkylated only at an unhindered primary amine group. A preselected degree of steric hindrance at amine groups near each end of the chain enables cyclization by the `ketoform synthesis` by reaction with a ketone in such a manner as to form a polysubstituted piperazinone ("PSP") ring which includes N atoms of proximate primary and secondary amine groups of the alkylated PAPA. The PSP so formed may then be reacted with a reactive triazine ring so that a PSP substituent is linked to the triazine ring through a single N atom and at least two C atoms, to form a 2-oxo-piperazinyl-triazine ("PIP-T"). Oligomers of the PIP-T may be prepared.Type: GrantFiled: February 19, 1982Date of Patent: October 30, 1984Assignee: The B. F. Goodrich CompanyInventors: John T. Lai, Pyong N. Son
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Patent number: 4479948Abstract: Hypotensively active triazino-(2,1-a)isoquinoline compounds having the ring system ##STR1## and methods of making and using such compounds.Type: GrantFiled: July 8, 1982Date of Patent: October 30, 1984Assignee: Hoechst AktiengesellschaftInventors: Bansi Lal, Adolf D'Sa, Alihussein N. Dohadwalla, Noel J. de Souza, Horst Dornauer
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Patent number: 4471417Abstract: Poly-bis-triazinylimides of the formula ##STR1## are prepared from bis-(2,4-dichloro-1,3,5-triazin-6-yl)imides and polyalkylpiperidylamines.They are used as light stabilizers for polymers.Type: GrantFiled: March 29, 1982Date of Patent: September 11, 1984Assignee: Hoechst AktiengesellschaftInventors: Hartmut Wiezer, Gerhard Pfahler
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Patent number: 4460404Abstract: Condensed ring aromatic ureas and isoureas are useful as plant growth regulants and as pre- and/or post-emergence herbicides.Type: GrantFiled: September 22, 1982Date of Patent: July 17, 1984Assignee: E. I. DuPont de Nemours and CompanyInventor: George Levitt
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Patent number: 4453971Abstract: N-(heterocyclicaminocarbonyl)arylsulfonamides, such as 3-isocyanato-N-[(4-methoxy-6-methyl-1,3,5-triazin-2-yl)aminocarbonyl]benze nesulfonamide or methyl [3-[[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]aminosulfonyl]phenyl] carbamate, are useful for the regulation of plant growth and as herbicides.Type: GrantFiled: September 22, 1982Date of Patent: June 12, 1984Assignee: E. I. Du Pont de Nemours and CompanyInventor: George Levitt
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Patent number: 4451400Abstract: Halogenophosphazenes of the formula ##STR1## in which n denotes 3 to 100, are reacted with alcohols or amines having polyalkylpiperidyl groups to give compounds which are suitable for stabilizing synthetic polymers and are distinguished by a very high migration resistance.Type: GrantFiled: May 7, 1982Date of Patent: May 29, 1984Assignee: Hoechst AktiengesellschaftInventor: Hartmut Wiezer
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Patent number: 4435401Abstract: 2,4-Diaminoquinazoline compounds of the formula ##STR1## or a pharmaceutically acceptable salt thereof wherein R is a pyrimidinyl, pyrazinyl, pyridazinyl or triazinyl group linked to the piperazine ring by one of its carbon atoms, and optionally substituted by hydroxy, halogen, alkyl, aralkyl, alkoxy, aralkoxy, alkylthio, aryl, aryloxy and certain amino groups; their use as an antihypertensive agent and pharmaceutical compositions containing them.Type: GrantFiled: December 23, 1981Date of Patent: March 6, 1984Assignee: Pfizer Inc.Inventors: Simon F. Campbell, Rhona M. Plews
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Patent number: 4417917Abstract: Certain benzene-1,2-disulfonic acid derivatives are useful as agricultural chemicals, and in particular as herbicides.Type: GrantFiled: October 20, 1981Date of Patent: November 29, 1983Assignee: E. I. Du Pont de Nemours and CompanyInventors: George Levitt, Richard F. Sauers
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Patent number: 4416817Abstract: Novel 3-methoxy-2-oxoazetidine derivatives, which are shown by the following formula ##STR1## wherein R.sub.1 is amino, acylated amino or protected amino, are of value as intermediates for the synthesis of useful compounds represented by the formula ##STR2## wherein R.sub.1 has the same meaning as defined above, as drugs in the treatment of bacterial infections.Type: GrantFiled: November 18, 1981Date of Patent: November 22, 1983Assignee: Takeda Chemical Industries, Ltd.Inventors: Taisuke Matsuo, Michihiko Ochiai
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Patent number: 4415570Abstract: Compounds useful in the treatment of rheumatism or allergic nephritis which have the formula ##STR1## wherein X is halogen, hydroxy, lower alkyl, lower alkenyl, lower alkoxy, nitro or amino;Y is hydrogen, halogen, hydroxy, lower alkyl, lower alkenyl, lower alkoxy, nitro or amino; andZ is mono-(lower alkyl)amino, di-(lower alkyl)amino, piperidino, piperazino, pyrrolidino, or morpholino.Type: GrantFiled: June 1, 1982Date of Patent: November 15, 1983Assignee: Nippon Shinyaku Co. Ltd.Inventors: Hiroshi Enomoto, Akira Nomura, Yoshiaki Aoyagi, Yoshihisa Shibata
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Patent number: 4412856Abstract: The novel compounds of the formula I are useful selective herbicides for postemergence application in crops of cereals, maize and rice.In formula I, ##STR1## A is an unsubstituted or substituted amino group, Q is a C.sub.2 -C.sub.6 alkylene bridge, Y is an oxygen or sulfur atom or an unsubstituted or substituted nitrogen atom, and Z is an unsubstituted or substituted phenyl, naphthyl or heterocyclic radical, which phenyl radical, containing the bridge member Y, can additionally carry one to four further substituents.Type: GrantFiled: May 22, 1981Date of Patent: November 1, 1983Assignee: Ciba-Geigy CorporationInventors: Hans-Georg Brunner, Rolf Schurter, Henry Szczepanski
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Patent number: 4406897Type: GrantFiled: July 6, 1981Date of Patent: September 27, 1983Assignee: William H. Rorer, Inc.Inventors: Henry F. Campbell, Thomas H. Scholz, George H. Douglas
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Patent number: 4400505Abstract: Compounds of the formula ##STR1## wherein at least one of the groups contains a 4-piperidinyl moiety are disclosed as light stabilizers for polymers.Type: GrantFiled: July 20, 1981Date of Patent: August 23, 1983Assignee: American Cyanamid CompanyInventors: Frank F. Loffelman, Thomas E. Brady
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Patent number: 4394506Abstract: N-(heterocyclicaminocarbonyl)arylsulfonamides in which the aryl radical is substituted in the 2-position by a carboxy radical, ester, thioester, or amide thereof; e.g. N-[(4,6-dimethylpyrimidin-2-yl)aminocarbonyl]-2-methoxycarbonylbenzenesulf onamide or N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-2-methoxycarbonylbenze nesulfonamide; are useful for the regulation of plant growth and as pre-emergence and post-emergence herbicides.Type: GrantFiled: November 30, 1979Date of Patent: July 19, 1983Assignee: E. I. Du Pont de Nemours and CompanyInventor: George Levitt
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Patent number: 4393060Abstract: N-substituted-diglycidyl-isocyanurates having the formula: ##STR1## wherein R represents a hydrocarbon-containing radical selected from the group consisting of alkyl, aryl, aralkyl, alkaryl and cycloalkyl, optionally containing:(a) heterocycles except epoxides, and unsaturation, and(b) substituents selected from the group consisting of halogen, hydroxyl, amino, N-substituted amino, mercapto, alkylmercapto, arylmercapto, alkylsulfoxy, arylsulfoxy, alkoxy, aryloxy and acyloxy,and R.sub.1 represents a member selected from the group consisting of hydrogen and alkyl having from 1 to 4 carbon atoms, as well as the method for preparing said N-substituted-diglycidyl-isocyanurates, therapeutic compositions with cytostatic action comprising said N-substituted-diglycidyl-isocyanurates, and a method of treatment of malignant neoplasias in warm-blooded animals by administering a therapeutically effective amount of said N-substituted-diglycidyl-isocyanurate.Type: GrantFiled: October 7, 1980Date of Patent: July 12, 1983Assignee: Henkel Kommanditgesellschaft auf AktienInventors: Herbert Fischer, Manfred Budnowski, Ulrich Zeidler
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Patent number: 4387225Abstract: Heterocyclic alkyl s-triazine compounds are prepared from the corresponding amidinourea and amidinothiourea compounds by reacting with an activated form of an acid amide to give respectively substituted s-triazinones and thiones of the formula ##STR1## which have pharmacological properties that render them suitable for use for a variety of medicinal purposes, including use as antidiarrheal agents, and which are also useful derivatives in analyzing for the corresponding amidinourea or amidinothiourea precursors.Type: GrantFiled: May 12, 1981Date of Patent: June 7, 1983Assignee: William H. Rorer, Inc.Inventors: George H. Douglas, William L. Studt, Chong M. Won, Stuart A. Dodson, Jerome J. Zalipsky
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Patent number: 4386177Abstract: Oligomers prepared from alkoxycarbonylalkyleneamino halotriazines and diamines are useful as light stabilizers for polymers subject to ultraviolet radiation degradation.Type: GrantFiled: July 20, 1981Date of Patent: May 31, 1983Assignee: American Cyanamid CompanyInventor: Frank F. Loffelman
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Patent number: 4356024Abstract: A process for the preparation of a 1-amino-1,3,5-triazine-2,4(1H, 3H)-dione compounds comprising the steps of reacting an N-substituted imido-dicarboxylic acid diaryl ester with an isothiosemicarbazone at a temperature of between 50.degree. and 150.degree. C. to form a 1-alkylidene-amino-1,3,5-triazine-2,4(1H, 3H)-dione reaction product; and thereafter, hydrolyzing the reaction product in an acid medium. The reaction product need not be separated from the reaction mixture before the hydrolysis step. Certain novel 1-amino-1,3,5-triazine-2,4(1H, 3H)-dione compounds are provided. The compounds are useful as herbicides.Type: GrantFiled: February 10, 1981Date of Patent: October 26, 1982Assignee: Bayer AktiengesellschaftInventors: Karlfried Dickore', Engelbert Kuhle
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Patent number: 4348493Abstract: Ultraviolet light stabilizers for polymers are disclosed.Type: GrantFiled: July 20, 1981Date of Patent: September 7, 1982Assignee: American Cyanamid CompanyInventor: Frank F. Loffelman
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Patent number: 4348219Abstract: Novel 2-[[(heterocyclic)-aminocarbonyl]aminosulfonyl]benzeneacetic acid derivatives, such as 2-[[(4,6-dimethoxypyrimidin-2-yl)-aminocarbonyl]aminosulfonyl]benzeneaceti c acid, methyl ester, are useful as plant growth regulants and herbicides.Type: GrantFiled: April 29, 1981Date of Patent: September 7, 1982Assignee: E. I. Du Pont de Nemours and CompanyInventor: George Levitt
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Patent number: 4331586Abstract: Oligomers of the formula ##STR1## which contain at least one piperidinyl moiety in the repeating unit are useful as light stabilizers for polymers.Type: GrantFiled: July 20, 1981Date of Patent: May 25, 1982Assignee: American Cyanamid CompanyInventor: William B. Hardy
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Patent number: 4329456Abstract: The present invention relates to a process for the preparation of vat dyes of the formula ##STR1## in which A is a vattable radical, X is an acyl radical and Y' is a halogen atom, an amino group or an aryloxy group, which comprises acylating compounds of the formula ##STR2## in which A is as defined under formula (1) and Y is a halogen atom, with an acylating agent which contains the acyl radical X, and, if desired, subjecting the compounds of the formula (2), before or after acylation, to a condensation reaction with an amine or an aromatic hydroxy compound.Type: GrantFiled: May 15, 1980Date of Patent: May 11, 1982Assignee: Ciba-Geigy AGInventor: Athanassios Tzikas
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Patent number: 4315859Abstract: Novel oligomer or polymer polyamine-1,3,5-triazines containing at least one polyalkylpiperidine radical, for example that of the formula ##STR1## processes for their production, their use for stabilizing organic material, and the organic material protected therewith against oxidative and light-induced degradation.Type: GrantFiled: January 4, 1980Date of Patent: February 16, 1982Assignee: Ciba-Geigy CorporationInventor: Erwin Nikles
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Patent number: 4310346Abstract: This invention relates to N(Substituted Phenylsulfonyl) N'(Substituted Pyrimidinyl) urea compounds having the formulae I and IA ##STR1## to agricultural compositions containing them and to their methods of use as general as well as selective pre- and post-emergence herbicides and as plant growth regulants.Type: GrantFiled: May 30, 1980Date of Patent: January 12, 1982Assignee: E. I. Du Pont de Nemours and CompanyInventors: George Levitt, Richard F. Sauers
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Patent number: 4302241Abstract: This invention relates to novel N-(heterocyclicaminocarbonyl)arylsulfonamides in which the aryl radical is substituted by two carboxyl radicals. The compounds have utility as herbicides.Type: GrantFiled: November 30, 1979Date of Patent: November 24, 1981Assignee: E. I. Du Pont de Nemours and CompanyInventor: George Levitt
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Patent number: 4301286Abstract: This invention relates to herbicidal O-alkyl sulfonylisoureas which are useful as herbicides, both general and selective.Type: GrantFiled: August 20, 1979Date of Patent: November 17, 1981Assignee: E. I. Du Pont de Nemours and CompanyInventors: Gregory W. Schwing, Thomas S. Woods
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Patent number: 4294963Abstract: Polyalkylpiperidine derivatives which are unsubstituted in the 1-position of the piperidine ring and in the 4-position are bonded through a heteroatom bridge to an s-triazine radical, can be converted by reaction with a dihalide or a di-, tri- or tetraepoxide into compounds of the formula I ##STR1## wherein n is 2, 3 or 4 and p is 0 or 1. Polymer or oligomer compounds of the formula II ##STR2## wherein n represents the degree of polymerization and E and E' represent end groups, are obtained by reacting a triazine derivative which contains at least two polyalkylpiperidine substituents with dihalides or diepoxides.Both types of compound are stabilizers for polymers, especially against damage by light. They are distinguished by low volatility and a low tendency to migrate, so that they are of special interest for use in thin polymer layers, for example in fibres, sheets or coatings.Type: GrantFiled: July 16, 1979Date of Patent: October 13, 1981Assignee: Ciba-Geigy CorporationInventor: Jean Rody
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Patent number: 4288593Abstract: Novel polyalkylpiperidine derivatives of s-triazines of the formula ##STR1## in which X and X' are a divalent organic radical, X", X.sub.1 and X.sub.2 are a direct bond or a divalent organic radical, Y, Y', Y", Y.sub.1, Y.sub.2, Z and Z' are --O--, --S--, --NH-- or --NR.sup.3 --, R is H or CH.sub.3 and R.sup.1, R.sup.2 and R.sup.3 are a monovalent organic radical or a polyalkylpiperidine group, or the group R.sup.1 --X"--Y"-- is chlorine, and R.sup.4 is H, O, alkyl, allyl or benzyl, are valuable stabilizers for polymeric materials, in particular to protect them against photochemical degradation. The derivatives are prepared by stepwise reaction of cyanuric chloride with the corresponding YH, Y'H and Y"H compounds.If 2 or 3 of these components are identical, the corresponding symmetrically substituted triazine compounds, which are preferred, are formed.Type: GrantFiled: January 28, 1980Date of Patent: September 8, 1981Assignee: Ciba-Geigy CorporationInventor: Jean Rody
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Patent number: 4287338Abstract: The present invention provides novel substituted sulfooxy-pyrimidinium, -pyridinium, and -triazinium hydroxide inner salts. These compounds are useful for the treatment of hypertension and peripheral vascular diseases. They are formed by reacting the corresponding aminopyrimidine, aminotriazine, and aminopyridine N-oxides with a latent sulfate source such as pyridinium-sulfur trioxide complex, triethylamine-sulfur trioxide complex, chlorosulfonic acid or chlorosulfuryl chloride.Type: GrantFiled: March 10, 1980Date of Patent: September 1, 1981Assignee: The Upjohn CompanyInventor: John M. McCall
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Patent number: 4281123Abstract: Three substituents are introduced into cyanuric acid in the presence of an acid binding agent by working in a manner permitting high mixing and therefore high reaction velocities and permitting high throughputs in small tubular containers by introducing liquid cyanuric chloride through a nozzle in the upper portion of the mixing apparatus in countercurrent flow to upwardly flowing reactants (and acid binding agent) introduced from at least one lower nozzle above a breast shaped constriction in the lower, open portion of the apparatus. The process can be carried out at normal, reduced or elevated pressure.Type: GrantFiled: November 16, 1979Date of Patent: July 28, 1981Assignee: Deutsche Gold- und Silber-Scheideanstalt vormals RoesslerInventors: Klaus Hentschel, Friedrich Bittner
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Patent number: 4281124Abstract: Compounds of the formula ##STR1## wherein E denotes a reactive substituent which can be split off,D denotes hydrogen, optionally substituted alkyl, aryl, aralkyl, aminocarbonyl, mono- or di-alkylaminocarbonyl, optionally substituted alkoxy, alkylthio, aryloxy, arylthio, aralkoxy or aralkylthio, or a radical of the formula ##STR2## G and G.sub.1 independently of one another denote hydrogen, optionally substituted alkyl, aryl or aralkyl, or, together with N, a 5-membered or 6-membered ring,B and B.sub.1 independently of one another denote a linking member--X--Y--Z--Y.sub.1 --whereinX is bonded to the triazine radical and denotes oxygen, sulphur or ##STR3## R denotes hydrogen, optionally substituted alkyl, alkenyl or aralkyl, Y denotes ##STR4## n denotes a number from 0 to 4, Z denotes an optionally substituted phenylene or naphthylene radical or the radical of the formula --CH.dbd.CH--,Y.sub.1 denotes a radical of the formula ##STR5## n.sub.1 denotes a number from 0 to 4, n and n.sub.Type: GrantFiled: November 29, 1979Date of Patent: July 28, 1981Assignee: Bayer AktiengesellschaftInventors: Bernd Berger-Lohr, Karl H. Schundehutte, Manfred Soll
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Patent number: 4275203Abstract: Chloro-amino-s-triazines are produced by the known reaction of cyanuric chloride with an amine or .alpha.-aminonitrile in the presence of an acid binding agent in an improved manner by working at high mixing velocities and thus at high reaction speed and thereby obtaining high throughputs in small tubular containers by introducing liquid cyanuric chloride through a nozzle in the upper portion of the mixing apparatus in countercurrent flow to upwardly flowing reactants (plus acid binding agent) introduced from at least one lower nozzle about a breast shaped constriction in the lower, open portion of the apparatus. The process can be carried out at normal, reduced or elevated pressure.Type: GrantFiled: November 16, 1979Date of Patent: June 23, 1981Assignee: Deutsche Gold und Silber Scheideanstalt vormals RoesslerInventors: Klaus Hentschel, Friedrich Bittner
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Patent number: 4261892Abstract: This disclosure describes new compounds and compositions of matter useful as anti-inflammatory agents and as inhibitors of the progressive joint deterioration characteristic of arthritic disease and the methods of meliorating inflammation and of inhibiting joint deterioration in mammals therewith, the active ingredients of said compositions of matter being certain 2,4,6-tris(substituted-amino)-s-triazines.Type: GrantFiled: March 5, 1979Date of Patent: April 14, 1981Assignee: American Cyanamid CompanyInventors: Andrew S. Tomcufcik, Adolph E. Sloboda
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Patent number: 4246409Abstract: Novel s-triazine compounds are prepared as derivatives of the corresponding amidinourea and amidinothiourea compounds by reacting with an activated form of an acid amide to give substituted s-triazinones and thiones respectively, of the formula ##STR1## The s-triazinones and thiones are useful derivatives in analyzing for the corresponding amidinourea or amidino thiourea precursors and also have useful pharmacological properties which make them suitable for a variety of medicinal purposes including use as antidiarrheal agents.Type: GrantFiled: November 13, 1978Date of Patent: January 20, 1981Assignee: William H. Rorer, Inc.Inventors: George H. Douglas, William L. Studt, Chong M. Won, Stuart A. Dodson, Jerome J. Zalipsky
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Patent number: 4237284Abstract: The present invention relates to reactive dye-compounds of formula I, ##STR1## in which Y is hydrogen or sulpho,X is a straight chain or branched (C.sub.2-6) alkylene group or ##STR2## in which each of A.sub.1 and A.sub.2, independently, is a direct bond or a (C.sub.1-4) alkylene group, n is 1 or 2 and the ring D is optionally substituted by up to three (C.sub.1-4) alkyl groups,with the proviso that when n is 2, the group ##STR3## is the radical of an unsymmetrical diamine, R.sub.1 is hydrogen; (C.sub.1-4) alkyl; (C.sub.2-4) alkyl substituted in the .beta.,.gamma.-or .delta.-position by hydroxy and/or carboxy; or (C.sub.5-6) cycloalkyl or (C.sub.1-4) alkyl-substituted (C.sub.5-6) cycloalkylZ is the radical of a fibre reactive group which contains a single fibre reactive componentor mixtures thereof, which compounds are in free acid or water-soluble salt form and are useful as dyestuffs for dyeing or printing hydroxy group-containing or nitrogen containing organic textile substrates.Type: GrantFiled: September 14, 1978Date of Patent: December 2, 1980Assignee: Sandoz Ltd.Inventor: Roland Mislin
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Patent number: 4228281Abstract: Dicarboxylic acids containing at least two triazine rings are very suitable for producing thermoplastic polyesters having high glass transition temperatures and high dimensional stability under heat, and at the same time good processing characteristics.Type: GrantFiled: September 18, 1978Date of Patent: October 14, 1980Assignee: Ciba-Geigy CorporationInventors: Thomas Kainmuller, Jurgen Habermeier, Lothar Buxbaum
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Patent number: 4225337Abstract: N-(heterocyclicaminocarbonyl)arylsulfonamides, such as 3-isocyanato-N-[(4-methoxy-6-methyl-1,3,5-triazin-2-yl)aminocarbonyl]benze nesulfonamide or methyl [3-[[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]aminosulfonyl]phenyl] carbamate, are useful for the regulation of plant growth and as herbicides.Type: GrantFiled: October 27, 1978Date of Patent: September 30, 1980Assignee: E. I. Du Pont de Nemours and CompanyInventor: George Levitt
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Patent number: 4160831Abstract: 2-Cyclopropylamino-4-formamidino-6-amino-s-triazine of the formula ##STR1## wherein R.sub.1 represents hydrogen, C.sub.1 -C.sub.4 -alkyl which is unsubstituted or substituted by lower alkoxy; or represents C.sub.3 -C.sub.4 -alkenyl, C.sub.3 -C.sub.4 -alkynyl, cyclopropyl, hydroxyl, methoxy or ethoxy,R.sub.2 represents hydrogen methyl or ethyl, orR.sub.1 and R.sub.2 together with the nitrogen atom to which they are attached represent a 5- or 6-membered heterocyclic ring which can contain a further nitrogen atom or an oxygen atom,R.sub.3 represents methyl or ethyl,R.sub.4 represents methyl or ethyl, andR.sub.5 represents hydrogen or methyl for combatting developmental stages of insects.Type: GrantFiled: January 16, 1978Date of Patent: July 10, 1979Assignee: Ciba-Geigy CorporationInventors: Verena Laanio, Hans U. Brechbuhler, Dagmar Berrer
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Patent number: 4160832Abstract: 2-Cyclopropylamino-4-formylamino-6-amino-s-triazines of the formula ##STR1## wherein R.sub.1 represents hydrogen, C.sub.1 -C.sub.4 -alkyl which is unsubstituted or substituted by lower alkoxy, or represents C.sub.3 -C.sub.4 -alkenyl, C.sub.3 -C.sub.4 -alkynyl, cyclopropyl, hydroxy, methoxy or ethoxy,R.sub.2 represents hydrogen, methyl or ethyl, orR.sub.1 and R.sub.2 together with the nitrogen atom to which they are attached represent a 5- or 6-membered heterocyclic ring which can contain a further nitrogen atom or an oxygen atom, andR.sub.3 represents hydrogen or methyl,And the acid addition salts thereof for combatting developmental stages of insects.Type: GrantFiled: January 16, 1978Date of Patent: July 10, 1979Assignee: Ciba-Geigy CorporationInventors: Verena Laanio, Hans U. Brechbuhler, Dagmar Berrer